Indications and side effects of the drug Riboxin in ampoules: instructions for use. "Riboxin": reviews of doctors and athletes How to take riboxin in bodybuilding

11.04.2022 Accessories

    Riboxin is a drug that improves the contractility of the heart, corrects its rhythm, reduces oxygen starvation of tissues and regulates the metabolism of the body.

    At its core, it is a source of energy for the myocardium and coronary vessels. In parallel, the drug prevents ischemia of the kidneys during surgery, participates in the metabolism of glucose and takes on the functions of ATP in its absence in the body. Adenosine triphosphate is present in every cell, but with age or disease, its amount decreases, which requires an additional source of energy supply from the outside.

    The use of Riboxin in sports is justified, since physical activity requires increased endurance, and this drug becomes an additional source of energy.

    Composition and forms of release

    Riboxin is available in tablets and ampoules for oral and injectable use. It is based on inosine, a metabolic stimulant that generates energy in the body. In addition, starch, methylcellulose, sucrose and other elements of the cachet are present as additional substances in the tableted version. The drug belongs to list B, that is, it is released only by prescription.

    As a source of energy, Riboxin is of interest to athletes who, during training, give themselves increased physical activity. The fact is that at the molecular level it is the basis for ATP (adenosine triphosphate) - the basis of the life of the body. The main function of this acid, which is produced independently in the body, is to maintain the optimal state of the heart muscle and guarantee the absence of hypoxia in the tissues.

    Riboxin becomes an additional substance that stops the lack of ATP in different situations. The drug is responsible for the correction of arrhythmias, accelerates, expands the coronaries, which stimulates the strength of heart contractions and improves blood flow.

    In practice, the patient experiences a surge of strength, chest pains, migraines, weakness, fatigue disappear, shortness of breath practically ceases to bother him.

    Riboxin is stored in a dark place, out of the reach of children, at a temperature of 0 to +25 degrees, for 5 years.

    ATP precursor

    Riboxin is sometimes called a vitamin for the heart. But this is not a very accurate definition. Indeed, without its main component - inosine - cells are not able to absorb either vitamins or trace elements. Hypoxia occurs in them, and the heart may even stop. Since inosine is a nucleoside that is part of every cell membrane, its deficiency provokes a violation of the functions of various organs and tissues. The first to suffer:

    • The cardiovascular system, in which ischemia, atherosclerosis, myocardial dystrophy progresses against the background of hypoxia.
    • The liver, oxygen starvation of which leads to inflammation with an outcome in cirrhosis. Hepatocytes suffer, iron loses its function as a natural filter.
    • Eyes, namely: the ophthalmic nerve and muscles of the eye apparatus. Loss of visual acuity and contrast.
    • Kidneys with the formation of uroporphyria - a metabolic disorder at the local level.
    • Stomach - hypoxic toxicosis violates the integrity of the mucosa with the formation of erosions.

    Riboxin, getting into the body, puts everything in its place. As a source of ATP, it reduces pressure, normalizing the vascular wall, but it turns out to be dangerous for hypotensive patients. It stimulates the immune system, helping to resist radiation therapy. The same properties of the drug are also used in sports to withstand the intensity of stress in training and competition, to prevent sprains of muscles and ligaments.

    Instructions for use

    Riboxin is taken according to certain rules.

    • If it is injected, and this is the most optimal delivery of inosine to the body, then intramuscular injections or intravenous administration are selected: drip or jet. The first injection is 200 mg once a day. In the absence of side effects, the dose is doubled. Course - 10 days. Through a dropper, the medicine is administered slowly to exclude heartbeat: no more than 50 drops per minute.
    • Tablets or capsules are used from the age of twelve. The first dose is a tablet (capsule) three times a day. With good tolerance, the dose is increased: first to two tablets three times a day, and then to four. Metabolic disorders change the scheme: one tablet 4 times a day, for a month or three. Reception takes place 30 minutes before meals, capsules are washed down with plain water.
    • For athletes, the best regimen is to take pills a couple of hours before training. The course is no more than three months with a break of 30 days. A side effect of Riboxin is the accumulation of muscle mass.

    Contraindications for admission

    A big plus of Riboxin is the minimum of contraindications. But they are:

    Body sensitization, urticaria. When the drug is discontinued, everything disappears.

    • Exacerbation of gout with prolonged oral administration. Purine, which is a precursor of Riboxin, is involved in the conversion of uric acid. Its prolonged presence in the body provokes an attack of gout.
    • Leukemia in the terminal stage.
    • Individual intolerance.
    • Prenatal weeks and the period of breastfeeding require minimization of the drug intake or its complete exclusion.

    In the case of chemotherapy, there is a danger of metabolic hyperuricemia with an outcome in gout. Therefore, oncologists prescribe the drug with great care and under close supervision.

    Pregnancy before prenatal weeks is not a restriction to taking Riboxin. On the contrary, he saves expectant mothers from many heart troubles. It also insures the progression or debut of gastritis, the pathology of the biliary system. A feature of the drug is its positive effect on the fetus, the prevention of its hypoxia. But Riboxin is prescribed only by a doctor, in dosages corresponding to the condition of the mother and fetus.

    Treatment of heart pathologies

    The heart muscle is constantly experiencing stress associated with ensuring normal nutrition and oxygen supply to tissues. With age, it wears out, that is, it becomes dependent on additional energy support. It is provided by Riboxin, which acts as a cardioprotector. It interrupts the chain of negative processes triggered by muscle ischemia, protecting myocardial cells.

    Unfortunately, its mechanism of action has not been thoroughly studied. But it is reliably known that, being a derivative of purine and a precursor of ATP, it exhibits the qualities of an anabolic. With its help, anaerobic glycolysis is activated, that is, anoxic energy production using glucose. This reduces its concentration in the myocardium and enables Riboxin to stimulate the synthesis of nucleotides and protein under ischemia, acting as a cardioprotector.

    This is how the metabolic potentiation of Riboxin manifests itself. This effect of the drug is used not only for the treatment of myocardial ischemia, but also for hypertension, arrhythmias.

    With hypertension

    In case of high pressure, Riboxin affects cell receptors, restoring their function. This is especially effective in the early stages of the disease. In parallel, the drug dissolves cholesterol plaques, which corrects the work of blood vessels and restores metabolism. In combination with Enapril, Renitek, Curantil, Delix, Enalzid and other hypotensive drugs that the doctor selects, this gives a good result. There is a long and persistent decrease in blood pressure.

    However, when using Riboxin in combination with other drugs, it should be remembered that it is not combined with certain medications, and if alcohol is consumed during treatment, it can lead to a hypertensive crisis or exacerbation of cardiac pathology.

    With arrhythmia

    Violation of the heart rhythm is clinically manifested by a change in the heart rate in one direction or another, dizziness, shortness of breath. As a rule, this is a secondary symptom of some underlying disease. Therefore, before building a treatment regimen, you need to accurately diagnose. However, Riboxin is the same drug, the appointment of which for arrhythmias of any genesis is indicated without fear of negative consequences. Especially effective is its use with potassium preparations.

    The essence of its action in arrhythmia is reduced to the normalization of metabolism in the heart muscle. Riboxin freely penetrates into each cell and, increasing its energy balance, restores the normal conduction of electrical impulses through the myocardium. This stops the arrhythmia.

    It should be noted that such a uniquely positive effect on the heart and blood vessels makes the drug indispensable in the complex therapy of cardiovascular pathology. Including during the acute phase of myocardial infarction.

    Recently, articles have appeared in medical journals that Riboxin is a placebo. However, practice says something completely different. Its action is confirmed by animal experiments and clinical trials.

    Treatment of the digestive system

    Riboxin is a derivative of purine. It is phosphorylated, penetrating into hepatocytes, and converted into inosinic acid. This substance is a source of nucleotides, both adenyl and guanyl, which are responsible for the functioning of the digestive system. Acquiring the properties of the curator of the gastrointestinal tract, the drug guarantees:

    • Optimization of energy-dependent reactions, creation of the basic basis for redox processes, formation of macroenergy molecules, stimulation of tissue respiration, lactate utilization. All this, as it were, duplicates the functions of the liver, removing part of the load from it.
    • Synthesis of a whole complex of purine nucleosides necessary for the formation of DNA and RNA. This stimulates regenerative processes in the food tube and aids in adaptive synthesis.

    In practice, biochemical transformations scientifically proven in laboratory conditions are visualized in the correction of metabolism, the removal of free radicals, the decrease in antitoxic function, and the rapid regeneration of liver tissue and gastric mucosa. Riboxin is indicated for hepatitis and cirrhosis of various genesis and at different stages of pathological inflammation.

    Compatibility with other tools

    Riboxin is absolutely incompatible with alcohol, especially when administered parenterally and with B vitamins, in particular B6. But it is combined without problems with almost all drugs that are prescribed for the treatment of diseases of the cardiovascular, digestive and urinary systems: Nitroglycerin, Concor, Renitek, Enapril, Nifedilin, Lazeks, Furosemide.

    The use of Riboxin in bodybuilding

    Understanding the benefits of additional energy that Riboxin brings to the body has led to its widespread use in power sports that require high energy consumption. The use of the drug allows:

    • Increase the concentration of hemoglobin in the blood to the optimal value, taking into account the throughput of the substance.
    • Stimulate the production of insulin by the pancreas, which ensures easy absorption of carbohydrates by the myocardium.
    • Adjust the lumen of the vessels depending on the voltage, increasing it.
    • Activate immunity.
    • Accelerate muscle regeneration.
    • Raise the level of endurance of the athlete.

    All this, especially endurance, is priceless for bodybuilding. In addition, Riboxin improves the blood supply to all organs, including those responsible for potency, which is important for men.

    The multi-vector nature of the drug allows you to completely stop energy costs when performing strength exercises, guaranteeing normal oxygen supply, and, therefore, respiration and tissue nutrition, that is, metabolism.

    At the same time, one should not forget about a sense of proportion and caution. That is, before using Riboxin, a complete clinical and laboratory examination is shown to assess the state of the body and its need for a drug. Athletes using Riboxin easily tolerate physiological hypoxia, since tissue cells absorb oxygen to the maximum. At the same time, the myocardium works calmly and confidently.

    The use of Riboxin in sports

    The popularity of Riboxin among athletes is by no means associated with the effect of losing weight, as is the case with many other drugs. Abroad, inosine is included in the menu of every athlete. This is due to the fact that it does not just normalize the work of the main internal organs: the heart. liver, kidneys, but also stimulates the body's defenses, forms a high endurance to macroloads.

    Since Riboxin is a complete analogue of inosine, it also acts: it strengthens the walls of blood vessels, prevents ruptures and sprains of muscles and ligaments. This is appreciated in any sport, but especially among the "siloviki". The indisputable advantage of the drug is that it meets all anti-doping requirements. In addition, it has been proven to be completely safe (with the exception of individual intolerance) and effective in the recovery of athletes after extreme physical exertion.

    Sports nutrition

    The most popular with Riboxin (inosine) are:

    • Premium Inosine from Ultimate Nutrition.
    • Inosine from Mega-Pro.
    • Inosine from Life Extension.
    • Cell-Tech Hardcore by MuscleTech.

As non-steroidal helpers. Riboxin is one of the very first and popular sports drugs. According to the main classification, it belongs to metabolic agents. Why is Riboxin used in bodybuilding? How to take, how much and what dosage to choose? All these questions are of interest to athletes who want to drink a course of the drug.

The purpose and benefits of Riboxin

Riboxin, or inosine, is a nucleic acid that has a purine base. Inosine is also a precursor of ATP, a substance directly involved in metabolic processes and the formation of energy for muscles. In medicine, it is usually used to improve cardiac activity, as well as stimulate the growth of new cells in damaged organs and tissues.

Riboxin effects in bodybuilding:

  • It has an antihypoxic property, that is, it enhances the protective properties of the body with a lack of oxygen. This is due to the effect of expanding blood vessels and increasing the throughput of hemoglobin when taking the drug;
  • Inosine is taken to increase immunity, which is especially important during heavy physical exertion;
  • Improves reparative processes, which allows you to recover faster after training;
  • Riboxin is taken to speed up metabolism, improve metabolism in the body;
  • Increases stamina - this makes it possible to increase the intensity of training.

Separately, it should be noted about the effect of inosine on the heart. After all, this muscle is severely tested in sports and is quickly depleted. It is useful to take Riboxin for the prevention of heart damage and with weakening of the myocardium, cardiac disorders, cardiomyopathy, angina pectoris.

It is customary to use the remedy for diseases and damage to the liver from taking pharmaceuticals, hepatitis, ulcers of the digestive system. Taking care of your health and the activity of vital organs will have a great effect on your athletic performance. It is also useful to take riboxin as a rehabilitation therapy after taking alcohol and steroid drugs.

For a long time it was believed that inosine would help and keep it dry. In addition, many bodybuilders have used the drug to increase weight and gain strength in training. However, modern research shows that Riboxin does not have anabolic properties, so it will not help to gain weight and become stronger.

Instructions for use Riboxin

Inosine is produced in the form of tablets and injections. The average cost of the drug is about 50 rubles, depending on the manufacturer, in one package there are usually 50 tablets. The price of inosine ampoules is slightly more expensive - from 70 rubles.

Riboxin is taken orally half an hour before a meal. The first four days should begin with small doses - no more than 0.8 g per day. In the future, if the drug is well tolerated by the body, the total dosage of inosine is 1.5-2 g, the maximum allowable dose is 2.5 g per day. It is recommended to use inosine - 3-4 times a day, approximately 2 tablets of 200 mg at a time. A more accurate dosage is calculated depending on the weight of the athlete - 0.15 g per 10 kg of weight.

The minimum duration of the course is 4 weeks, the maximum is 3 months. Particular attention should be paid to taking Riboxin on training days and immediately before training.

What non-steroidal drugs go well with Riboxin in bodybuilding? These are vitamin-mineral complexes, B vitamins, adaptogens. They should also be consumed in courses for 1-2 months, and then take a long break. Potassium orotate should be taken one hour before meals or a couple of hours after, 0.5 g 4 times a day. When taking orotate and riboxin, it is better to drink them with a break of half an hour, but there will be nothing wrong if you take pills from different drugs at the same time.

Good day, comrades! Today I want to touch on the so-called topic. That is, those funds that are popular in the ranks of naturally engaged athletes who want to improve their athletic performance. After all, few are ready to go on.

And I understand these people one hundred percent! In search of effective drugs, athletes, as a rule, turn their eyes towards non-steroidal anabolic agents. The most popular among them is Riboxin. Today we will talk about how effective Riboxin is in bodybuilding.

Riboxin (inosine) is a metabolic agent that, in simple terms, “improves the formation of new structures in the body.” In the case of this drug, energy characteristics are improved, due to its effect on the formation of ATP (the main source of energy). Inosine affects the coronary circulation and metabolic processes in the myocardium, resulting in a beneficial effect on the heart muscle. Participates in the supply of muscle tissue with oxygen.

For some effects Riboxin. The latter, in turn, has been actively used by our athletes for recovery, since the days of the USSR, until the World Anti-Doping Agency (WADA) added it to the list of prohibited substances.

Riboxin has also been used in sports since the distant 70s. But recent studies have questioned its effectiveness, so the popularity of the drug has declined somewhat.

However, many experienced athletes, including bodybuilding representatives, use this drug.

Why is Riboxin needed in bodybuilding?

Why do athletes use this tool?

First of all, due to its anabolic action. Since the drug is a precursor of ATP and promotes the formation of this energy compound. As a consequence, this leads to an increase in explosive power. After all, ATP is used by our body in the first few seconds of intensive work with iron.

Due to its ability to deliver oxygen to the muscles, the drug should improve aerobic capacity.

It makes sense to take Riboxin during intense loads, which occur during the period of preparation for competitions or when the load on the heart increases due to growing body weight.

Inosine is also needed for recovery after a course of anabolic steroids, as it has hepatoprotective properties (positively affects liver function). And as you know, the liver suffers from taking certain steroid drugs. But ruthless research, as always, casts a shadow of doubt on its effectiveness. So the choice of whether or not to take the drug is yours alone.

Instructions for use

Before proceeding to the instructions for use, I will say a few words about the forms of release of the drug.

Riboxin is available in the form of tablets and injections. It is not recommended to administer the drug intramuscularly. Perhaps with intramuscular injection there will be a better effect of the drug, since you bypass the gastrointestinal tract. But is it worth it? - I doubt.

Now let's talk about how to take the drug.

Riboxin is recommended to be taken before meals. The dosage in bodybuilding is 1.5 - 2.5 grams per day. Start with a daily dose of 0.6 - 0.8 grams 3 - 4 times a day. If the drug is well tolerated, then increase the dose to 2.5 grams. The duration of the course is 1-2 months.

Many bodybuilders recommend taking Riboxin with Asparkam. Since it supplies the heart and muscles with such important elements as potassium and magnesium. Often their deficiency leads to muscle cramps. Therefore, during intense training, it is advisable to take these two drugs in conjunction. A more expensive analogue of Asparkam is Panangin.

In pharmacies, you can now find the drug Asparkam Avexima, which is several times more expensive than regular Asparkam. Aveksima is a Russian manufacturer. The active ingredients are the same - potassium and magnesium, but the more expensive drug gets better reviews. Despite the fact that it is more expensive than Asparkam, it still costs less than Panangin.

Another agent used in conjunction with Riboxin is Potassium orotate. But its intake is justified only in case of a lack of potassium in the body, which can be expressed by muscle weakness, a drop in blood pressure and muscle spasms.

Contraindications and side effects

The drug should not be taken if you have intolerance to the active substance - inosine or its other components. In the presence of gout, Riboxin is also not recommended. As with problems with the metabolic processes of uric acid and purine bases in the body.

It is forbidden to use inosine together with alcohol. Since such a bundle can cause serious complications.

Side effects, in the absence of contraindications, are rare. But with prolonged use, it should be borne in mind that the drug increases the concentration of uric acid in the blood. In some cases, possible: bradycardia (low pulse), itching and redness of the skin (as a result of hyperemia).

Despite the seeming harmlessness, the drug can be dangerous when used independently. Therefore, I strongly recommend that you consult with a specialist before starting the reception!

Accept or not?

Riboxin, despite studies that deny its effectiveness in sports, is still used by athletes in many countries. On sports forums, this drug is one of the most discussed among nonsteroidal drugs. Moreover, a large number of people leave positive feedback about the effect of inosine on the body,.

In any case, if you decide to take this drug, be sure to consult a specialist!

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Consider one of the nutritional supplements commonly used in sports - riboxin. It is mainly used by other athletes who are trying to keep their body in perfect condition. This food supplement is also called Inosine.

What does it look like?

Riboxin for athletes has the form of an odorless white powder, which has a bitter taste and cannot be dissolved in water.

Action on the body

After using this supplement, you feel a surge of energy, it speeds up metabolism and supplies all human organs with oxygen. Let's take a closer look at how Riboxin acts on the body:

  • improves metabolic processes in the body;
  • affects the synthesis of proteins, which is simply necessary for athletes;
  • promotes the formation of ATP;
  • does not allow oxygen starvation in the body;
  • increases blood flow;
  • fills the whole body with energy;
  • improves heart function;
  • helps to get rid of gastritis during pregnancy.

By using this nutritional supplement, athletes can spend a lot of time in the gym and feel very good. The drug Riboxin is recommended for use for the heart, as well as after drinking.

How to take Riboxin for athletes?

The daily dose of this dietary supplement is 1.5-2 g, if you translate this into tablets, then this is 7-14 pcs. It is necessary to use it before meals, 4 times a day. It is not necessary to take Riboxin before training, since the total amount of the dose taken before meals will be enough. First, to get used to the body, drink 1 tablet at a time, and then gradually increase your dose to 3 pcs. The duration of taking this dietary supplement is a maximum of 3 months, after which it is necessary to take a break of about 2 months.

Side effects

We figured out how to take Riboxin in sports, now let's look at possible side effects.

In general, there are no violations, unless you have intolerance to the supplement, kidney failure or gout. If you exceed the dose, then you may experience the following disorders: Allergy in the form of a rash on the skin, which may itch and peel off. The heartbeat may also be disturbed and heaviness in the chest may be felt.

In sports, Riboxin will help you achieve excellent results and form a beautiful body relief. Thanks to nutritional supplements and enhanced training, you can achieve the desired result.

In the Soviet Union in the 70s, the Riboxin drug was popular among weightlifters.

There was no official confirmation that it provides high results in sports, and for some time it was forgotten.

Today, at the second peak of popularity, Riboxin is actively used in strength sports, for which it is used - we will figure it out in this article.

Description and release form

The drug is a non-steroidal anabolic agent, which athletes take in combination with the course. In power sports, anabolics serve to strengthen bone and muscle tissues, their growth and renewal. Abroad, it is better known as inosine. At its core, it is a nucleic acid that stimulates the production of proteins and the synthesis of purines, maintaining the energy balance of cells. In medicine, it is used as a drug to prevent ischemia.

The product is available in tablets or injections, also in the form of an auxiliary component in additives -. In tablets, these are blisters with capsules of 0.2 g of inosine, 10, 20, 30, 40, 50 pieces each. In injections, a two percent solution of ten ampoules per pack, ampoules of 5 ml and 10 ml.

Did you know? The father of bodybuilding is considered to be Evgeny Sandov, who in 1901 organized the first performance of athletes who trained according to his own methodology. Eugene Sandow himself in 1894 became a world record holder, having squeezed out a bar with a weight of 122 kg with one hand.

Impact on the body of athletes

Those who take Riboxin have activated metabolism and, due to this, the lack of oxygen during exercise does not cause discomfort. A positive effect is observed on the muscle, which is important during physical exertion, especially in powerlifting.

The agent is actively involved in the metabolic process of glucose in the body, oxidative and reduction processes, improves tissue respiration. By increasing the strength of contractions of the heart muscle, it helps to relax the myocardium, improves blood circulation and blood supply to tissues.

The use of the drug prevents platelets from sticking together (which leads to the formation of blood clots), activates the ability of cells and tissues to regenerate.


To summarize, the use of the drug by athletes gives the following results:
  • Increases elasticity.
  • The level and throughput of hemoglobin is maintained.
  • The synthesis of insulin is normalized.
  • Stimulates digestibility.
As a result, after all of the above, the protective function of the body increases in athletes. Recent studies have not revealed any positive effect of the drug directly on or on the athlete's strength indicators, therefore, they will be effective for muscle building, and the drug will help to cope with severe ones, thereby increasing their effectiveness.

Important! Riboxin, like any drug, must be safe for the health of athletes, so before taking the remedy, it is advisable to consult a specialist doctor.


Indications for use

In medicine, the drug is prescribed for the treatment of cardiovascular diseases, the drug improves coronary circulation. It is prescribed for diseases of the stomach, duodenum. As an adjuvant that improves the function of the optic nerve, in combination with the treatment of glaucoma.

It is used as a means of supporting the heart muscle, it is especially recommended to take during the "drying". The drug by its action protects the muscles and ligaments from sprains and complications associated with them.

So, indications for use in sports:

  • Prevention of metabolic damage (MCD) of the myocardium during extreme physical exertion.
  • Prevention of cardiac arrhythmias.
  • Violation of carbohydrate, protein and fat metabolism.
  • Non-inflammatory myocardial damage due to heavy loads.
  • Liver damage after taking medications.
  • , acute and chronic hepatitis.
  • Ulcer of the stomach and duodenum.

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Methods of application and doses

The answer to the question: how to take Riboxin in tablets depends on the indications for use. In bodybuilding, to strengthen the heart muscle and greater endurance during exercise, take the drug three times a day, half an hour before meals, at a dosage of 1.5-2.5 g.

Reception begins in small doses from 0.6-0.8 grams three times a day or 0.2 grams four times a day. In the absence of negative effects, the dosage is increased. The course of admission is from four weeks to three months.

Injections in sports are used extremely rarely and not for body structure, but more for medical reasons.

Side effects and overdose

Contraindication is the drug, as well as renal failure. In case of an overdose, bradycardia (cardiac arrhythmias) and hyperemia (impaired blood flow), itching, uric acid concentration in the blood, skin flushing (redness in some areas) are possible. In the presence of gout, prolonged use in large doses will lead to an exacerbation of the disease.

In bodybuilding and powerlifting, taking the drug allows you to achieve maximum results, due to an increase in endurance during intense training. The body of an athlete under heavy loads is protected from injuries and quickly recovers.